Introduction
Anpiraterone acetate yog ib qho inhiben synthemes uas tuaj yeem tsim 17 - hydroxylase / C17,20-Lyase (CYP17).
Cov lus qhia
USP
Tshuaj lom neeg npe
(3) -17- (3-pyridinyl) androsta-5,16-dien-3-ol acetate.
Molecular Cov Qauv
C26H33Tsis muaj2
Cas tsis muaj.
154229-18-2
Yam ntim
1kg / tin
Daim ntawv muaj cai
sssssss
Hom
Anti - mob cancer
Chaw ntim khoom
Khaws rau hauv qhov tsaus ntuj thiab ua kom nws kaw.
Kev taw tes
Nws yog tsuas yog siv nyob rau hauv kev sib xyaw nrog prednisone lossis prednisone acetate rau kev kho mob ntawm Metastatic Castration (MRPC) Nws kuj tau qhia rau kev kho mob ntawm cov neeg mob siab- kev pheej hmoo, tsis muaj kev pheej hmoo ua ke nrog and}}}} kev kho mob.
Chaw muag khoom Cov Khoom Siv
Chav Tshuaj hauv Chav:Nws yog Cytochrome P 450 17 A1 (Cyp17A1) Inhibitor.
Mechanism ntawm Kev Ua:Anpiraterone acetate yog metabolized hauv vivo rau abiraterone, uas xaiv Inhibits CYP17A1. Cov enzyme no koom nrog hauv Biosynthesis ntawm androgens hauv cov kev xeem, cov qog adrenal, thiab prostate cancer hlwb. Los ntawm inhibiting cyp17a1, abiraterone acetate txo cov kab mob androgens, yog li kev txhawb nqa prostate lawv xav tau kev loj hlob thiab muaj peev xwm loj hlob.
Muab thiab tswj hwm
Cov tshuaj pom zoo ntawm abiraterone acetate yog 1000 mg (plaub {}} mg ntsiav tshuaj) ib zaug txhua hnub, noj tshuaj. Nws yuav tsum tau noj ntawm lub plab khoob, tsawg kawg 1 teev ua ntej lossis 2 teev tom qab noj mov. Prednisone lossis prednisone acetate feem ntau tau noj conmomitantly, ntawm ib koob ntawm 5 mg ob zaug ib hnub. Txoj kev kho yuav tsum txuas ntxiv mus kom txog thaum kab mob zuj zus lossis tsis tsim nyog muaj tshuaj lom. Txawm li cas los xij, cov tshuaj ntau thiab kev kho mob tshwj xeeb tuaj yeem hloov kho raws li tus neeg mob tus mob thiab teb rau kev kho.
Phiv thiab cov kev sib raug zoo
Cov kev mob tshwm sim ntau
Cov no suav nrog kev ua kom nkees, sib koom ua noj, Edema, cov pa dej kub, raws plab, hnoos, thiab cov mob tso zis.
Kev phiv loj
Qee qhov kev mob tshwm sim hnyav yuav tshwm sim, xws li mob siab lom, uas tuaj yeem ua kom daim siab ua kom lub siab enzyme, Jaundice, thiab muaj mob hnyav, mob siab ua tsis tiav. Muaj kuj muaj kev pheej hmoo ntau ntawm cov xwm txheej plawv Ib qho ntxiv, tsis muaj peev xwm tshwm sim, tshwj xeeb tshaj yog thaum cov tshuaj siv hauv kev sib xyaw nrog corticosteroids, xav tau kev saib xyuas zoo thiab tswj hwm qhov tsim nyog.
Cim npe nrov: ABIRILERONE ACETATE, Tuam Tshoj Abiraterone Acetate Manufacturers, lwm tus neeg, Hoobkas
